Protein Details: P2X receptor B

Protein ID

ICDB_Pro_0970

Protein Name

P2X receptor B

Gene Name

p2xB; DDB_G0275293

Organism

Dictyostelium discoideum (Social amoeba)

Length

369 amino acids

AlphaFoldDB

AF-Q553Y1-F1-model_v4.pdb

Function

P2X receptors are ATP-gated ion channels that play a role in intracellular calcium signaling. Not required for the purinergic response to extracellular nucleotides. Not essential for osmoregulation. Inward currents are evoked by intracellular ATP and ATP analogs. Insensitive to the P2 receptor antagonists PPADS and suramin; and also copper ions. Inhibited by sodium ions. Permeable to chloride ions.

Sequence

MTIDWDSILSYNTIKVVRIRDRRLGILHLCFLIVIVLYVVVYSAIIKKGYVTTEEPVGSIRTSLLAPDELKSNQAYCKNNTEPYPYEKLDCVYYDEKLALFPIGDDVGFTASTRMRISDQTVNCSLMNPSCKFYTNTSMNVYLADIESFTVLIDHTMYAPSSQIQFNGDDLSGYVLDQNGNEIQLNESVNTIGVQGKPDILQLGKLLEFAGVDLDGPSLVNSSNSIRYDGCVLFVFIEYSNTFSYDLKKIKYVYSIKKVDDTAYDVPEVIILNNENSRLYYKRHAIRLIFIQTGVIGSFNFQSLLLTLVSGLGLLTVSTLIVDQLAIRFLPQRKSYSSLKFQTTESFRMKKKIVNDDGEDKLYHNIEAL

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

Disease

Location

DOI ID

10.1038/nature00847; 10.1038/nature03481; 10.1074/jbc.m109.045674

RefSeq

XP_643830.2

Feature